SCHEMBL8928241

SCHEMBL8928241

CC1=C(C#N)C(c2cccc(-n3ccnc3)c2)C(C(=O)OC(C)C)=C(C)N1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.53
NR3C2 P08235 3/20 0.52
NR1I2 O75469 1/20 0.47
NR3C1 P04150 1/20 0.47
ABCB1 P08183 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
TBXA2R P21731 1/20 0.47
AGTR1 P30556 1/20 0.47
CCKBR P32239 1/20 0.47
PTGS2 P35354 1/20 0.47
PDE4D Q08499 1/20 0.47
SCN5A Q14524 1/20 0.47
SLC29A1 Q99808 1/20 0.47
CACNA1C Q13936 5/20 0.44
CACNA1F O60840 2/20 0.44
CACNA1D Q01668 2/20 0.44
CACNA1S Q13698 2/20 0.44
MEN1 O00255 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8928277 0.88 CACNA1C (0.54) NR3C2ADORA3CACNA1CCACNA1FCACNA1D
SCHEMBL8928204 0.87 CACNA1C (0.40) KDM4EPDE4DCACNA1CLMNAMAPT
SCHEMBL8860432 0.84 POLB (0.49) KDM4ECYP1A2CYP3A4CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL8928281 0.84 POLB (0.48) KDM4ECYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10475638 0.82 CACNA1F (0.50) KDM4ENR3C2ADORA3CACNA1CCACNA1F
SCHEMBL30357940 0.80 CACNA1F (0.54) KDM4EADORA3CACNA1CCACNA1FCACNA1D
SCHEMBL7269131 0.80 CACNA1F (0.54) KDM4EADORA3CACNA1CCACNA1FCACNA1D
SCHEMBL7268117 0.78 IDO1 (0.47) PDE4DCYP3A4
SCHEMBL10475641 0.78 ADORA3 (0.47) NR3C2ADORA3CACNA1CCACNA1FCACNA1D
SCHEMBL7277695 0.78 CACNA1C (0.48) KDM4EADORA3CACNA1CCACNA1FCACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP claimed
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP disclosed