SCHEMBL8928258

SCHEMBL8928258

CCOC(=O)c1c(C)nc(C)c(C#N)c1-c1cccc(-n2ccnc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.51
L3MBTL1 Q9Y468 3/20 0.51
SMN1; SMN2 Q16637 4/20 0.49
KDM4E B2RXH2 4/20 0.47
HPGD P15428 3/20 0.47
GAA P10253 3/20 0.47
LMNA P02545 3/20 0.47
MAPT P10636 3/20 0.47
NPSR1 Q6W5P4 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
HTT P42858 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
POLB P06746 1/20 0.40
MITF O75030 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
MAPK1 P28482 1/20 0.37
FNTA P49354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8928263 0.84 ALDH1A1 (0.52) ALDH1A1L3MBTL1SMN1; SMN2KDM4EHPGD
SCHEMBL8928275 0.84 CYP3A4 (0.49) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL6137231 0.80 ALDH1A1 (0.60) ALDH1A1L3MBTL1SMN1; SMN2KDM4EHPGD
SCHEMBL6137171 0.78 ALDH1A1 (0.58) ALDH1A1L3MBTL1SMN1; SMN2KDM4EHPGD
SCHEMBL6137339 0.77 ALDH1A1 (0.56) ALDH1A1L3MBTL1SMN1; SMN2KDM4EHPGD
SCHEMBL6137255 0.76 SMN1; SMN2 (0.56) ALDH1A1L3MBTL1SMN1; SMN2KDM4EHPGD
SCHEMBL6137213 0.74 ALDH1A1 (0.54) ALDH1A1L3MBTL1SMN1; SMN2KDM4EHPGD
SCHEMBL6137355 0.73 ALDH1A1 (0.56) ALDH1A1L3MBTL1SMN1; SMN2KDM4EHPGD
SCHEMBL4081415 0.73 L3MBTL1 (0.58) ALDH1A1L3MBTL1SMN1; SMN2KDM4ELMNA
SCHEMBL27740113 0.72 ALDH1A1 (0.42) ALDH1A1L3MBTL1KDM4EHPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP claimed
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP disclosed