SCHEMBL8928407

SCHEMBL8928407

CCc1cc2c(s1)-n1c(C)nnc1CN=C2c1ccccc1F

nearest known ligand 0.79

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.79
PDE4D Q08499 1/20 0.79
PTAFR P25105 18/20 0.59
GABRA1 P14867 1/20 0.54
GABRA5 P31644 1/20 0.54
GABRA2 P47869 1/20 0.54
GABRB2 P47870 1/20 0.54
CYP3A4 P08684 1/20 0.53
ALOX15 P16050 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Etizolam SCHEMBL42920 0.88 OPRK1 (1.00) OPRK1PDE4DPTAFRCYP3A4ALOX15
Etizolam SCHEMBL30665015 0.88 OPRK1 (1.00) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928436 0.86 OPRK1 (0.77) OPRK1PDE4DPTAFRGABRA1GABRA5
SCHEMBL11508119 0.85 PTAFR (0.65) OPRK1PDE4DPTAFRGABRA1GABRA5
Etizolam SCHEMBL28142121 0.84 OPRK1 (0.69) OPRK1PDE4DPTAFRGABRA1GABRA5
Etizolam SCHEMBL10869413 0.84 OPRK1 (0.90) OPRK1PDE4DPTAFRCYP3A4ALOX15
Etizolam SCHEMBL28086661 0.81 OPRK1 (0.85) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8928483 0.80 OPRK1 (0.84) OPRK1PDE4DPTAFRCYP3A4ALOX15
SCHEMBL8878960 0.80 OPRK1 (0.74) OPRK1PDE4DPTAFRGABRA1GABRA5
SCHEMBL8928481 0.79 OPRK1 (0.84) OPRK1PDE4DPTAFRCYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0776892-A1 THIENYLAZOLE COMPOUND AND THIENOTRIAZOLODIAZEPINE COMPOUND YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-06-04 EP disclosed