SCHEMBL8941845

SCHEMBL8941845

FC(F)(F)Sc1ccc(Cl)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.58
KDM4E B2RXH2 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
PTPRZ1 P23471 4/20 0.50
PTPN1 P18031 2/20 0.50
MAPT P10636 2/20 0.50
NPSR1 Q6W5P4 2/20 0.50
KCNK2 O95069 2/20 0.45
KCNK10 P57789 2/20 0.45
LMNA P02545 2/20 0.42
CYP2A6 P11509 1/20 0.42
HTT P42858 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
KIF11 P52732 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8005997 0.84 KCNK2 (0.54) ALDH1A1KDM4ETDP1PTPRZ1MAPT
SCHEMBL8941503 0.80 LMNA (0.38) ALDH1A1KDM4ETDP1PTPRZ1PTPN1
SCHEMBL13950430 0.80 MAPT (0.41) ALDH1A1KDM4ETDP1PTPRZ1PTPN1
SCHEMBL10935258 0.79 ALDH1A1 (0.58) ALDH1A1KDM4ETDP1PTPRZ1PTPN1
SCHEMBL25118409 0.78 MAPT (0.37) ALDH1A1KDM4ETDP1PTPRZ1PTPN1
SCHEMBL7940607 0.76 ALDH1A1 (0.61) ALDH1A1KDM4ETDP1PTPRZ1PTPN1
SCHEMBL10978325 0.76 ALDH1A1 (0.61) ALDH1A1KDM4ETDP1PTPRZ1PTPN1
SCHEMBL12436758 0.75 MAOA (0.44) ALDH1A1KDM4ETDP1PTPRZ1PTPN1
SCHEMBL28540817 0.75 ALDH1A1 (0.40) ALDH1A1KDM4ETDP1PTPRZ1PTPN1
SCHEMBL16555940 0.75 ALDH1A1 (0.43) ALDH1A1KDM4ETDP1PTPRZ1PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3632892-B1 METHOD FOR PRODUCING 3-ARYLPROPIONAMIDE COMPOUND SUMITOMO CHEMICAL CO (JP) 2024-07-31 EP disclosed
CN-110799490-B 3-arylpropionamide compound and method for producing 3-arylpropionate compound 住友化学株式会社 2023-05-02 CN disclosed
US-11028056-B2 Method for producing 3-arylpropionamide compound and 3-arylpropionic acid ester compound SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2021-06-08 US disclosed
US-20200165209-A1 METHOD FOR PRODUCING 3-ARYLPROPIONAMIDE COMPOUND AND 3-ARYLPROPIONIC ACID ESTER COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2020-05-28 US disclosed
EP-3632892-A1 METHOD FOR PRODUCING 3-ARYLPROPIONAMIDE COMPOUND AND 3-ARYLPROPIONIC ACID ESTER COMPOUND Sumitomo Chemical Company, Limited (JP) 2020-04-08 EP disclosed
CN-110799490-A Process for producing 3-arylpropionamide compound and process for producing 3-arylpropionate compound 住友化学株式会社 2020-02-14 CN disclosed
CN-110372550-A Aryl ether and application thereof 佩洛通治疗公司 2019-10-25 CN disclosed
CN-105530923-B Aryl ethers and their use 佩洛通治疗公司 2019-07-23 CN disclosed
WO-2015168368-A1 FLUOROALKYLATION REAGENTS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2015-11-05 WO disclosed
WO-2015168368-A1 FLUOROALKYLATION REAGENTS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2015-11-05 WO disclosed
US-4446078-A REACTING A POLYHALOALKOXY- OR POLYHALOALKYLTHIOBENZENE WITH A CARBOXYLIC DERIVATIVE, BORON TRIFLUORIDE RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1984-05-01 US disclosed
US-4438043-A Process for preparation of di- or trifluoromethoxyphenyl ketones or di- or trifluoromethylthiophenyl ketones RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1984-03-20 US disclosed
EP-0023422-B1 HERBICIDAL SULFONAMIDES, PREPARATION AND USE THEREOF, AND COMPOSITIONS CONTAINING THEM E.I. DU PONT DE NEMOURS AND COMPANY (US) 1984-02-22 EP disclosed
US-4431808-A ANTIDEPRESSANTS; TRANQUILIZERS; NEUROLEPTIC AGENTS SPOFA, SPOJENE PODNIKY PRO ZDRAVOTNICKOU VYROBU (CS) 1984-02-14 US disclosed
EP-0092627-A1 Process for the preparation of di- or trifluoromethoxyphenyl ketones or of di- or trifluoromethylthiophenyl ketones RHONE-POULENC CHIMIE (FR) 1983-11-02 EP disclosed
EP-0085265-A1 Process for the preparation of alpha,alpha-difluoroalkoxy or alpha,alpha-difluoroalkylthiophenyl ketones RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1983-08-10 EP disclosed
EP-0084743-A1 Process for the preparation of alpha, alpha-difluoroalkoxy or alpha, alphadifluoroalkylthiophenyl sulfones RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1983-08-03 EP disclosed
EP-0064322-A2 Benzenesulfonyl isocyanates, isothiocyanates, chlorides, and sulfonamides having a fluorinated substituent E.I. DU PONT DE NEMOURS AND COMPANY (US) 1982-11-10 EP disclosed
EP-0023422-A2 Herbicidal sulfonamides, preparation and use thereof, and compositions containing them E.I. DU PONT DE NEMOURS AND COMPANY (US) 1981-02-04 EP disclosed
US-4020169-A FROM ARYL IODIDE OR BROMIDE AND TRIFLUOROMETHYL THIO COPPER MERCK & CO., INC. (US) 1977-04-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200165209-A1 METHOD FOR PRODUCING 3-ARYLPROPIONAMIDE COMPOUND AND 3-ARYLPROPIONIC ACID ESTER COMPOUND AADAC, DDT, NAT1 ALDH1A1 116/4885KDM4E 1788/4885TDP1 1825/4885
US-11028056-B2 Method for producing 3-arylpropionamide compound and 3-arylpropionic acid ester compound AADAC, DDT, NAT1 ALDH1A1 116/4885KDM4E 1788/4885TDP1 1825/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.