SCHEMBL8942307

SCHEMBL8942307

NC(=O)NCCN(O)C(=O)c1ccc(Oc2ccccc2)o1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 1/20 0.43
ALDH1A1 P00352 3/20 0.41
MAPT P10636 2/20 0.41
NPSR1 Q6W5P4 2/20 0.40
MAPK1 P28482 2/20 0.39
ALOX5 P09917 3/20 0.36
PLAAT3 P53816 2/20 0.36
PLAAT5 Q96KN8 2/20 0.36
PLAAT2 Q9NWW9 2/20 0.36
PLAAT4 Q9UL19 2/20 0.36
NPC1 O15118 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35
TSHR P16473 1/20 0.35
ALOX12 P18054 1/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
EPHX2 P34913 3/20 0.34
LTA4H P09960 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8942702 0.88 EPHX2 (0.38) KLKB1ALDH1A1MAPTMAPK1ALOX5
SCHEMBL8942311 0.88 ALOX5 (0.49) ALDH1A1MAPTALOX5EPHX2LTA4H
SCHEMBL8942383 0.88 ALDH1A1 (0.45) ALDH1A1MAPTNPSR1MAPK1ALOX5
SCHEMBL8782994 0.85 KLKB1 (0.48) KLKB1ALDH1A1MAPTNPSR1MAPK1
SCHEMBL8942484 0.80 PARP10 (0.50) ALDH1A1ALOX5NPC1HPGDRAB9A
SCHEMBL8942399 0.78 CTNNB1 (0.52) ALDH1A1MAPTNPSR1MAPK1HPGD
SCHEMBL8783508 0.75 ALOX5 (0.54) ALDH1A1MAPTALOX5
SCHEMBL8783029 0.75 ALDH1A1 (0.50) KLKB1ALDH1A1MAPTNPSR1MAPK1
SCHEMBL8782600 0.75 KLKB1 (0.44) KLKB1ALDH1A1MAPTALOX5HPGD
SCHEMBL4155326 0.74 PARP10 (0.50) KLKB1ALDH1A1MAPTNPSR1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5514702-A Arylamidoalkyl-N-hydroxyurea compounds having lipoxygenase inhibitory activity ABBOTT LABORATORIES (US) 1996-05-07 US disclosed