SCHEMBL8945799

SCHEMBL8945799

CNC(Cc1ccccc1N)c1csc(Cl)n1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
YTHDC1 Q96MU7 1/20 0.33
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
HIF1A Q16665 1/20 0.31
HSD17B10 Q99714 1/20 0.31
LTA4H P09960 1/20 0.31
SLC6A3 Q01959 1/20 0.31
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945959 0.85 HDAC1 (0.35) CYP2C19LTA4HSLC6A3
SCHEMBL8945988 0.79 YTHDC1 (0.33) YTHDC1MEN1NPC1ALDH1A1CYP1A2
SCHEMBL8946086 0.78 RAD52 (0.41) NPC1ALDH1A1CYP3A4RAB9ABACE1
SCHEMBL8946109 0.76 YTHDC1 (0.32) YTHDC1
SCHEMBL8945955 0.73 TSHR (0.38) ALDH1A1CYP1A2CYP3A4CYP2D6SLC6A3
SCHEMBL8946074 0.71 AR (0.34)
SCHEMBL8945905 0.71 YTHDC1 (0.33) YTHDC1
SCHEMBL8945903 0.71 LTA4H (0.36) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9001661 0.70 ALDH1A1 (0.42) ALDH1A1
SCHEMBL8946115 0.70 SLC6A2 (0.31) SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed