SCHEMBL8945888

SCHEMBL8945888

Cc1ccsc1C(Cc1cc(Br)ccc1N)N(C)C

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KRAS P01116 1/20 0.33
ALOX5 P09917 1/20 0.33
S100B P04271 1/20 0.31
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945876 0.81 ALOX5 (0.35) ALOX5SLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL9425401 0.80 MAPT (0.30) ALOX5
SCHEMBL8946066 0.70 ALOX5 (0.33) ALOX5
SCHEMBL8945857 0.69 ALDH1A1 (0.32) ALOX5ALDH1A1
SCHEMBL8945773 0.68 CXCR1 (0.33) ALOX5ALDH1A1
SCHEMBL8945840 0.68 ALOX5 (0.35) ALOX5ALDH1A1
SCHEMBL8946090 0.68 ALOX5 (0.39) ALOX5ALDH1A1
SCHEMBL10409265 0.67 KDM4E (0.37) SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8946088 0.67 ALOX5 (0.41) ALOX5ALDH1A1
SCHEMBL8945834 0.67 MAPT (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed