SCHEMBL8945946

SCHEMBL8945946

COc1ccccc1CC(c1sccc1C)N(C)C=O

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
HTT P42858 1/20 0.38
HPGD P15428 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
AOC3 Q16853 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
MAPK8 P45983 1/20 0.34
TNF P01375 1/20 0.34
NOD1 Q9Y239 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946005 0.83 ALOX5 (0.32) MEN1KMT2A
SCHEMBL8945840 0.83 ALOX5 (0.35) MEN1KMT2A
SCHEMBL8945985 0.83 RECQL (0.36) HTTCYP2D6MEN1KMT2A
SCHEMBL8946039 0.81 CXCR1 (0.32) KMT2A
SCHEMBL9425099 0.80 ALOX5 (0.33) KMT2A
Hydrochloric Acid SCHEMBL8945763 0.79 CXCR1 (0.32) KMT2A
SCHEMBL8946053 0.74 HPGD (0.40) HPGDCYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL9425592 0.73 KDM4E (0.31) KDM4EHPGD
Hydrochloric Acid SCHEMBL8945983 0.73 CYP2D6 (0.42) HPGDCYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL8945969 0.69 OPRM1 (0.44) POLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed