SCHEMBL8946961

SCHEMBL8946961

COc1ccc2[nH]c(I)c(CCN)c2c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 6/20 0.72
HTR1D P28221 5/20 0.72
TSHR P16473 3/20 0.63
CYP1A2 P05177 2/20 0.63
MTNR1A P48039 2/20 0.63
MTNR1B P49286 2/20 0.63
CYP3A4 P08684 1/20 0.63
CYP2D6 P10635 1/20 0.63
CYP2C9 P11712 1/20 0.63
NQO2 P16083 1/20 0.63
CYP2C19 P33261 1/20 0.63
ALDH1A1 P00352 5/20 0.59
HTR1A P08908 4/20 0.54
HTR7 P34969 4/20 0.54
MAPT P10636 4/20 0.54
HTR2A P28223 3/20 0.54
TRPM8 Q7Z2W7 2/20 0.54
HTR2C P28335 2/20 0.54
NFKB1 P19838 1/20 0.54
HTR1B P28222 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25969437 0.87 MTNR1A (0.64) HTR6HTR1DTSHRCYP1A2MTNR1A
SCHEMBL4244966 0.84 HTR1D (1.00) HTR6HTR1DTSHRCYP1A2MTNR1A
SCHEMBL8229569 0.82 HTR6 (0.72) HTR6HTR1DTSHRCYP1A2MTNR1A
Hydrochloric Acid SCHEMBL7433474 0.82 HTR1D (0.97) HTR6HTR1DTSHRCYP1A2MTNR1A
SCHEMBL8691195 0.81 HTR6 (0.71) HTR6HTR1DTSHRCYP1A2MTNR1A
SCHEMBL8947088 0.81 HTR6 (0.73) HTR6HTR1DCYP1A2MTNR1AMTNR1B
SCHEMBL8947058 0.80 HTR6 (0.68) HTR6HTR1DTSHRCYP1A2MTNR1A
Cyanide SCHEMBL28561862 0.80 HTR1D (0.92) HTR6HTR1DTSHRCYP1A2MTNR1A
SCHEMBL25969475 0.79 TSHR (0.56) HTR6HTR1DTSHRCYP1A2MTNR1A
SCHEMBL2403262 0.78 HTR1D (0.65) HTR6HTR1DTSHRCYP1A2MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5552428-A ANTIARRHYTHMIA AGENTS FOR CARDIOVASCULAR DISORDERS USING MELATONIN DERIVATIVES INSTITUTO FARMACOLOGICO LOMBARDO-IFLO, S.A.S. (IT) 1996-09-03 US disclosed