SCHEMBL8948003

SCHEMBL8948003

CCCN(CCC)CCc1cc2sc(=O)n(CCN3CCC(C(=O)c4ccc(F)cc4)CC3)c2cc1OC

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.44
HTR2C P28335 2/20 0.44
DRD2 P14416 1/20 0.44
CNR2 P34972 2/20 0.42
HTR7 P34969 1/20 0.42
HTR6 P50406 1/20 0.42
WNT3A P56704 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
GRM2 Q14416 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948061 0.85 SIGMAR1 (0.52) HTR2AHTR2CCNR2HTR7HTR6
SCHEMBL8948024 0.85 HTR2A (0.47) HTR2AHTR2CDRD2CNR2HTR7
SCHEMBL8948001 0.84 HTR2A (0.43) HTR2AHTR2CDRD2CNR2HTR7
SCHEMBL8948051 0.79 HTR2A (0.55) HTR2AHTR2CDRD2HTR7HTR6
SCHEMBL8948150 0.79 HTR2A (0.55) HTR2AHTR2CDRD2CNR2HTR7
SCHEMBL8948058 0.77 CNR2 (0.49) HTR2AHTR2CDRD2CNR2HTR7
SCHEMBL8948000 0.75 HTR2A (0.50) HTR2AHTR2CDRD2HTR7HTR6
SCHEMBL8948034 0.75 HTR2A (0.52) HTR2AHTR2CDRD2CNR2HTR7
SCHEMBL8948192 0.75 HTR1A (0.65) HTR2AHTR2CHTR7GRM2
SCHEMBL8948121 0.74 HTR2A (0.57) HTR2AHTR2CDRD2HTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed