SCHEMBL8949037

SCHEMBL8949037

CCOC(=O)COC1CCCN(c2ccc(-c3ccc(C#N)cc3)nn2)C1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.41
RAB9A P51151 2/20 0.41
DGAT2 Q96PD7 3/20 0.40
DRD4 P21917 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.36
USP14 P54578 1/20 0.36
SCD O00767 1/20 0.36
GPBAR1 Q8TDU6 1/20 0.35
HRH2 P25021 1/20 0.35
HRH1 P35367 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8949331 0.75 NPC1 (0.41) NPC1RAB9ADGAT2MAPTSCD
SCHEMBL8949168 0.72 ITGB3 (0.43) NPC1RAB9AMAPTSCD
SCHEMBL8948657 0.70 GRM2 (0.47) DRD4TMEM97SIGMAR1USP14
Hydrochloric Acid SCHEMBL8949350 0.69 NPC1 (0.42) NPC1RAB9AMAPTSCDHRH3
SCHEMBL1742211 0.67 HTR6 (0.46) NPC1HRH2HRH1HRH3
SCHEMBL16128015 0.66 ALDH1A1 (0.52) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL8949328 0.66 ITGB3 (0.47) NPC1RAB9ASCD
SCHEMBL14587568 0.65 SMN1; SMN2 (0.52) ALDH1A1HRH3
SCHEMBL8770620 0.65 ITGB3 (0.55) KDM4EALDH1A1HRH2HRH1
SCHEMBL29852501 0.65 KDM4E (0.49) NPC1RAB9AKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed