SCHEMBL8951806

SCHEMBL8951806

COc1ccc(CC2C3CCCCC3CCN2C=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.43
HRH3 Q9Y5N1 2/20 0.37
EPHX2 P34913 2/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2066096 0.82 OPRK1 (0.43) OPRK1HRH3
SCHEMBL8951802 0.71 ALDH1A1 (0.37) HRH3ALDH1A1CYP3A4CYP2D6CYP2C19
SCHEMBL12859662 0.68 ALDH1A1 (0.54) EPHX2ALDH1A1KMT2ACYP2D6CYP2C9
SCHEMBL2064253 0.68 ALDH1A1 (0.54) EPHX2ALDH1A1KMT2ACYP2D6CYP2C9
SCHEMBL8477000 0.67 CYP3A4 (0.39) HRH3ALDH1A1CYP3A4CYP2D6CYP2C19
SCHEMBL3365060 0.66 LTA4H (0.51) HRH3EPHX2
SCHEMBL6628369 0.64 LTA4H (0.54) HRH3EPHX2
SCHEMBL28728795 0.64 SIGMAR1 (0.56) KMT2A
SCHEMBL11768994 0.64 HRH3 (0.46) HRH3HPGD
SCHEMBL11760698 0.64 HRH3 (0.46) HRH3HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5512577-A Bicyclic hexahydroaporphine and 1-benzyloctahydroisoquinoline therapeutic compositions and processes for utilizing said compositions CREIGHTON UNIVERSITY (US) 1996-04-30 US disclosed