SCHEMBL895863

SCHEMBL895863

Cc1ccc(C(=O)[C@H](C)N2CCCC2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 12/20 0.65
SLC6A2 P23975 11/20 0.65
CHRNB4 P30926 6/20 0.65
CHRNA3 P32297 6/20 0.65
SLC6A4 P31645 5/20 0.65
CHRNB2 P17787 5/20 0.65
CHRNA4 P43681 5/20 0.65
CHRNA1 P02708 4/20 0.65
CHRNG P07510 4/20 0.65
CHRNB1 P11230 4/20 0.65
CHRND Q07001 4/20 0.65
ALDH1A1 P00352 3/20 0.59
KDM4E B2RXH2 1/20 0.59
GAA P10253 1/20 0.59
CHRM2 P08172 1/20 0.58
ADRA2B P18089 1/20 0.58
DRD3 P35462 1/20 0.58
SIGMAR1 Q99720 1/20 0.58
HRH3 Q9Y5N1 1/20 0.58
LMNA P02545 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17644179 1.00 SLC6A3 (0.65) SLC6A3SLC6A2CHRNB4CHRNA3SLC6A4
Hydrochloric Acid SCHEMBL17645636 0.98 SLC6A3 (0.63) SLC6A3SLC6A2CHRNB4CHRNA3SLC6A4
SCHEMBL7946750 0.86 SLC6A3 (0.60) SLC6A3SLC6A2CHRNB4CHRNA3SLC6A4
SCHEMBL5813245 0.85 RAB9A (0.53) SLC6A3SLC6A2CHRNB4CHRNA3SLC6A4
SCHEMBL5954545 0.84 SLC6A3 (0.66) SLC6A3SLC6A2CHRNB4CHRNA3SLC6A4
SCHEMBL9597385 0.84 SLC6A3 (0.61) SLC6A3SLC6A2CHRNB4CHRNA3SLC6A4
SCHEMBL6811754 0.84 ALDH1A1 (0.61) SLC6A3SLC6A2CHRNB4CHRNA3SLC6A4
SCHEMBL11037118 0.84 SLC6A2 (0.67) SLC6A3SLC6A2CHRNB4CHRNA3SLC6A4
SCHEMBL28360223 0.84 SLC6A2 (0.67) SLC6A3SLC6A2CHRNB4CHRNA3SLC6A4
SCHEMBL9796926 0.83 SLC6A3 (0.60) SLC6A3SLC6A2CHRNB4CHRNA3SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8793078-B2 Method for predicting activation energy using atomic fingerprint descriptor or atomic descriptor BIOINFORMATICS & MOLECULAR DESIGN RESEARCH CENTER (KR) 2014-07-29 US disclosed
US-20120084012-A1 METHOD FOR PREDICTING ACTIVATION ENERGY USING ATOMIC FINGERPRINT DESCRIPTOR OR ATOMIC DESCRIPTOR BIOINFORMATICS & MOLECULAR DESIGN RESEARCH CENTER (KR) 2012-04-05 US disclosed
US-20110213558-A1 METHOD FOR PREDICTING ACTIVATION ENERGY USING AN ATOMIC FINGERPRINT DESCRIPTOR OR AN ATOMIC DESCRIPTOR BIOINFORMATICS & MOLECULAR DESIGN RESEARCH CENTER (KR) 2011-09-01 US disclosed
EP-2354987-A2 METHOD FOR PREDICTING ACTIVATION ENERGY USING AN ATOMIC FINGERPRINT DESCRIPTOR OR AN ATOMIC DESCRIPTOR Bioinformatics&Molecular Design Research Center (KR) 2011-08-10 EP disclosed
WO-2010056053-A2 METHOD FOR PREDICTING ACTIVATION ENERGY USING AN ATOMIC FINGERPRINT DESCRIPTOR OR AN ATOMIC DESCRIPTOR 사단법인 분자설계연구소 (KR) 2010-05-20 WO disclosed