SCHEMBL8959690

SCHEMBL8959690

COc1cn(CCN)c2ccc(F)cc12

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.51
GSK3B P49841 4/20 0.42
KDR P35968 2/20 0.41
FLT3 P36888 1/20 0.41
ICMT O60725 3/20 0.41
SLC6A2 P23975 3/20 0.38
SLC6A4 P31645 3/20 0.38
SLC6A3 Q01959 3/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38
DRD3 P35462 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ADRB2 P07550 1/20 0.37
CCNT1 O60563 1/20 0.36
CDK9 P50750 1/20 0.36
BRD4 O60885 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8959605 0.89 HTR6 (0.48) HTR6GSK3BKDRFLT3ICMT
Fumaric Acid SCHEMBL8959622 0.89 HTR6 (0.48) HTR6GSK3BKDRFLT3ICMT
SCHEMBL23927897 0.75 HTR3A (0.36) HTR6ICMTHTR2A
SCHEMBL23927894 0.75 HTR3A (0.36) HTR6ICMTHTR2A
SCHEMBL29780354 0.75 HTR3A (0.36) HTR6ICMTHTR2A
SCHEMBL8959806 0.72 HTR2A (0.40) HTR6GSK3BKDRFLT3HTR2A
SCHEMBL8959614 0.72 ICMT (0.39) ICMT
SCHEMBL12613820 0.70 HTR6 (0.61) HTR6KDM4EALDH1A1ADRB2
SCHEMBL29324209 0.70 HTR6 (0.50) HTR6GSK3BICMTHTR2A
SCHEMBL5785762 0.69 HTR6 (0.67) HTR6KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655440-A2 1-Aminoethylindoles F. HOFFMANN-LA ROCHE AG (CH) 1995-05-31 EP claimed
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
EP-0655440-A2 1-Aminoethylindoles F. HOFFMANN-LA ROCHE AG (CH) 1995-05-31 EP disclosed