SCHEMBL8965986

SCHEMBL8965986

CN(C)c1cccc(COc2ccc(N)nn2)c1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 10/20 0.52
NOS2 P35228 5/20 0.52
APP P05067 1/20 0.42
EGFR P00533 1/20 0.40
FFAR1 O14842 1/20 0.39
FYN P06241 1/20 0.38
ALDH1A1 P00352 2/20 0.37
TSHR P16473 1/20 0.37
BCAT2 O15382 1/20 0.36
PLK1 P53350 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8966289 0.86 THRA (0.44) NOS1NOS2FFAR1ALDH1A1BCAT2
SCHEMBL15618237 0.85 NOS1 (0.44) NOS1NOS2APPEGFRFYN
SCHEMBL8965946 0.81 IDO1 (0.51) FFAR1ALDH1A1
SCHEMBL8965939 0.79 MAOB (0.55)
SCHEMBL8965693 0.78 CYP3A4 (0.51)
SCHEMBL8965857 0.78 NUDT1 (0.43) NOS1NOS2APPFFAR1ALDH1A1
SCHEMBL933699 0.77 BCAT2 (0.55) ALDH1A1BCAT2
SCHEMBL4383894 0.72 IDO1 (0.58) ALDH1A1TSHR
SCHEMBL8965867 0.72 FFAR1 (0.38) NOS1FFAR1ALDH1A1BCAT2
SCHEMBL8965593 0.71 NOS1 (0.45) NOS1NOS2ALDH1A1BCAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5538970-A Treatment of cancer with imidazo-1,2-pyridazin compounds GLAXO WELLCOME INC. (US) 1996-07-23 US disclosed
US-5447956-A Anticarcinogenic agents BURROUGHS WELLCOME CO. (US) 1995-09-05 US disclosed
US-5380759-A Methyl N-[6-(3,4,5-trimethoxybenzloxy)imidazo[1,2-b]pyridazin-2-zyl]carbamate used to treat leukemia BURROUGHS WELLCOME CO. (US) 1995-01-10 US disclosed
EP-0305093-B1 Imidazo(1,2-b)pyridazine derivatives WELLCOME FOUND (GB) 1994-04-06 EP disclosed
US-5091531-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1992-02-25 US disclosed
EP-0305093-A1 Imidazo(1,2-b)pyridazine derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1989-03-01 EP disclosed