SCHEMBL8965693

SCHEMBL8965693

Nc1ccc(OCc2cccc(Cl)c2)nn1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.51
IDO1 P14902 2/20 0.51
AGXT P21549 2/20 0.51
MAOB P27338 3/20 0.51
GRM5 P41594 4/20 0.49
DHFR P00374 2/20 0.49
MPO P05164 2/20 0.48
DCPS Q96C86 1/20 0.47
PIN1 Q13526 1/20 0.46
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.45
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
RXRG P48443 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8965946 0.82 IDO1 (0.51) IDO1MAOBPIN1
SCHEMBL933699 0.80 BCAT2 (0.55) IDO1AGXTMAOB
SCHEMBL8965939 0.79 MAOB (0.55) IDO1AGXTMAOBMPOPIN1
SCHEMBL5026708 0.79 CYP3A4 (0.51) CYP3A4IDO1AGXTMAOBGRM5
SCHEMBL8965857 0.78 NUDT1 (0.43)
SCHEMBL8965986 0.78 NOS1 (0.52)
SCHEMBL8966289 0.76 THRA (0.44) CYP3A4MAOB
SCHEMBL21383991 0.73 PNMT (0.47) CYP3A4IDO1AGXTMPO
SCHEMBL30701931 0.73 NPC1 (0.67) CYP3A4IDO1AGXTMAOBGRM5
SCHEMBL29442787 0.73 PNMT (0.47) CYP3A4IDO1AGXTMPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5538970-A Treatment of cancer with imidazo-1,2-pyridazin compounds GLAXO WELLCOME INC. (US) 1996-07-23 US disclosed
US-5447956-A Anticarcinogenic agents BURROUGHS WELLCOME CO. (US) 1995-09-05 US disclosed
US-5380759-A Methyl N-[6-(3,4,5-trimethoxybenzloxy)imidazo[1,2-b]pyridazin-2-zyl]carbamate used to treat leukemia BURROUGHS WELLCOME CO. (US) 1995-01-10 US disclosed
US-5371219-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1994-12-06 US disclosed
EP-0305093-B1 Imidazo(1,2-b)pyridazine derivatives WELLCOME FOUND (GB) 1994-04-06 EP disclosed
US-5091531-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1992-02-25 US disclosed
EP-0305093-A1 Imidazo(1,2-b)pyridazine derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1989-03-01 EP disclosed