SCHEMBL8968172

SCHEMBL8968172

CC(C)(C)c1ccc(C#N)cc1NC(=O)Nc1cnccn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.52
NPC1 O15118 3/20 0.52
KDM4E B2RXH2 9/20 0.49
POLB P06746 2/20 0.49
MAPT P10636 2/20 0.49
PRKD3 O94806 3/20 0.47
MAP4K4 O95819 3/20 0.47
CLK2 P49760 3/20 0.47
GSK3A P49840 3/20 0.47
GSK3B P49841 3/20 0.47
LIMK1 P53667 3/20 0.47
CDK5 Q00535 3/20 0.47
DYRK1A Q13627 3/20 0.47
CLK4 Q9HAZ1 3/20 0.47
CDK1 P06493 2/20 0.47
CDK2 P24941 2/20 0.47
FLT4 P35916 2/20 0.47
CSNK1D P48730 2/20 0.47
CSNK2A1 P68400 2/20 0.47
STK3 Q13188 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8968165 0.85 NPC1 (0.52) RAB9ANPC1MAPTMEN1KMT2A
SCHEMBL8968218 0.81 CYP11B1 (0.54) RAB9ANPC1KDM4EMAPTMEN1
SCHEMBL8968747 0.81 CXCR1 (0.49) RAB9AKDM4EPOLBMAPTMEN1
SCHEMBL8970501 0.80 CXCR1 (0.45) RAB9ANPC1KDM4EPOLBMAPT
SCHEMBL8968160 0.75 CXCR2 (0.65) RAB9ANPC1KDM4EPOLBMAPT
SCHEMBL5381046 0.71 KDM4E (0.69) RAB9ANPC1KDM4EPOLBMAPT
SCHEMBL8968156 0.69 GAA (0.49) KDM4EPOLBGSK3BHTTHSD17B10
SCHEMBL8968199 0.69 ABCC9 (0.45) RAB9ANPC1MAPTMEN1KMT2A
SCHEMBL8968203 0.69 ABCC9 (0.45) RAB9ANPC1MAPTMEN1KMT2A
SCHEMBL3145830 0.69 P2RY1 (0.71) KDM4EMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0656350-A1 Biaryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1995-06-07 EP claimed
US-5547966-A Aryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1996-08-20 US disclosed
EP-0656350-A1 Biaryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1995-06-07 EP disclosed