SCHEMBL8968165

SCHEMBL8968165

CC(C)(C)c1ccc(C#N)cc1NC(=O)Nc1ccccn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.52
RAB9A P51151 6/20 0.52
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
MAPT P10636 1/20 0.49
FLT3 P36888 2/20 0.47
ADORA3 P0DMS8 1/20 0.47
PIM1 P11309 1/20 0.47
ADORA2A P29274 1/20 0.47
ADORA2B P29275 1/20 0.47
ADORA1 P30542 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PIM3 Q86V86 1/20 0.47
AURKB Q96GD4 1/20 0.47
MAPK13 O15264 1/20 0.47
MAPK12 P53778 1/20 0.47
MAPK11 Q15759 1/20 0.47
MAPK14 Q16539 1/20 0.47
GRIK1 P39086 1/20 0.46
LMNA P02545 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8968172 0.85 RAB9A (0.52) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL8968160 0.81 CXCR2 (0.65) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL8968747 0.79 CXCR1 (0.49) RAB9AMEN1KMT2AMAPTSMN1; SMN2
SCHEMBL8968218 0.78 CYP11B1 (0.54) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL17079609 0.77 RAB9A (0.69) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL17079611 0.76 GRM4 (0.67) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL8970501 0.76 CXCR1 (0.45) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL8968156 0.75 GAA (0.49) SMN1; SMN2MAPK13MAPK12MAPK11MAPK14
SCHEMBL8968189 0.73 ALDH1A1 (0.43) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL9750118 0.72 NPC1 (0.81) NPC1RAB9AMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547966-A Aryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1996-08-20 US claimed
EP-0656350-A1 Biaryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1995-06-07 EP claimed
US-5547966-A Aryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1996-08-20 US disclosed
EP-0656350-A1 Biaryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1995-06-07 EP disclosed