SCHEMBL8969096

SCHEMBL8969096

N=c1c2c(C(F)(F)F)cccc2nc2n1C1CC3CC(CC2C3)C1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
XPO1 O14980 2/20 0.36
HRH3 Q9Y5N1 2/20 0.33
ACHE P22303 1/20 0.33
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32
PDE10A Q9Y233 1/20 0.32
KCNH2 Q12809 3/20 0.31
GRM2 Q14416 2/20 0.31
HRH4 Q9H3N8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969453 0.84 ACHE (0.45) HRH3ACHECHRNB2CHRNA4
SCHEMBL8969422 0.82 HRH4 (0.34) ACHEHRH4
SCHEMBL8970053 0.81 ACHE (0.38) ACHE
SCHEMBL8968188 0.81 ACHE (0.32) ACHE
SCHEMBL8969708 0.81 ALDH1A1 (0.38) HRH3CHRNB2CHRNA4PDE10AKCNH2
SCHEMBL8968293 0.73
SCHEMBL8968811 0.73 LRRK2 (0.38) HRH3CHRNB2CHRNA4KCNH2
SCHEMBL8968897 0.71 BCHE (0.31) ACHE
SCHEMBL8969437 0.71 BCHE (0.35) ACHE
SCHEMBL8968356 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed