SCHEMBL8969708

SCHEMBL8969708

N=c1c2cccc(C(F)(F)F)c2nc2n1C1CC3CC(CC2C3)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NCF1 P14598 1/20 0.34
KCNH2 Q12809 5/20 0.33
HRH3 Q9Y5N1 1/20 0.33
PDE10A Q9Y233 1/20 0.33
ESR1 P03372 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32
ADORA2A P29274 5/20 0.32
ADORA1 P30542 5/20 0.32
CYP3A4 P08684 3/20 0.32
ADORA3 P0DMS8 2/20 0.32
ADORA2B P29275 1/20 0.32
CYP2C19 P33261 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NR1I2 O75469 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8968721 0.85 KDM4E (0.38) ALDH1A1L3MBTL1KDM4ELMNATSHR
SCHEMBL8969949 0.81 HRH4 (0.32) ALDH1A1CYP2C19
SCHEMBL8968606 0.81 ACHE (0.39) KCNH2HRH3ADRA1APARP1
SCHEMBL8969096 0.81 XPO1 (0.36) KCNH2HRH3PDE10ACHRNB2CHRNA4
SCHEMBL8968811 0.73 LRRK2 (0.38) KCNH2HRH3CHRNB2CHRNA4HTR2B
SCHEMBL8969661 0.69 BCHE (0.34) ALDH1A1L3MBTL1KDM4ELMNATSHR
SCHEMBL8969422 0.69 HRH4 (0.34) PARP1
SCHEMBL8970437 0.68 MPO (0.36)
SCHEMBL8969453 0.68 ACHE (0.45) HRH3CHRNB2CHRNA4PARP1
SCHEMBL8969462 0.68 PIK3CD (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed