SCHEMBL8969440

SCHEMBL8969440

CNC(=O)Oc1ccc2c(c1)CN1C(=N2)C2CC3CC(C2)CC1C3

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE P22303 10/20 0.38
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
HSD17B10 Q99714 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
BACE1 P56817 1/20 0.35
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
BCHE P06276 2/20 0.34
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
KMT2A Q03164 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8968787 0.86 ACHE (0.41) ACHEALDH1A1KDM4EHSD17B10SMN1; SMN2
SCHEMBL8969231 0.82 MAOA (0.35) ACHE
SCHEMBL8968566 0.80 ACHE (0.32) ACHEALDH1A1KDM4ESMN1; SMN2
SCHEMBL8968545 0.78 ACHE (0.39) ACHEALDH1A1KDM4EHSD17B10SMN1; SMN2
SCHEMBL8969986 0.78 MAOA (0.35) ACHEALDH1A1KDM4ESMN1; SMN2PDE3B
SCHEMBL8968791 0.76 HTR2A (0.34) PDE3BPDE3A
SCHEMBL9381793 0.76 ACHE (0.40) ACHEALDH1A1KDM4ESMN1; SMN2OPRM1
SCHEMBL8968314 0.75 PDE3B (0.40) ACHEPDE3BPDE3A
SCHEMBL8968336 0.74
SCHEMBL8969521 0.71 CTSD (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
EP-0597956-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1994-05-25 EP disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed