SCHEMBL8969478

SCHEMBL8969478

COc1cccc2c1OC(C(=O)NCCc1ccccc1)CC2

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.51
ATM Q13315 1/20 0.49
HPGD P15428 2/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 2/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
KDM4E B2RXH2 1/20 0.45
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TP53 P04637 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
ACHE P22303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969209 0.79 MEN1 (0.65) TAAR1HPGDMEN1KMT2AALDH1A1
SCHEMBL7552940 0.79 LTB4R (0.47) NFKB1NFKB2RELACA1CA2
SCHEMBL7552930 0.79 LTB4R (0.47) NFKB1NFKB2RELACA1CA2
SCHEMBL7557806 0.79 LTB4R (0.47) NFKB1NFKB2RELACA1CA2
SCHEMBL7319517 0.78 NFKB1 (0.52) HPGDNFKB1NFKB2RELACYP3A4
Hydrochloric Acid SCHEMBL8858324 0.78 LTB4R (0.47) NFKB1NFKB2RELACA1CA2
SCHEMBL8858322 0.75 MTNR1A (0.45) NFKB1NFKB2RELACA1CA2
SCHEMBL7314503 0.74 TDP1 (0.56) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL9379902 0.72 MTNR1A (0.45) NFKB1NFKB2RELACA1CA2
SCHEMBL24700600 0.72 TAAR1 (0.50) TAAR1ATMALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585392-A TREATING OR PREVENTING STROKES BAYER AKTIENGESELLSCHAFT (DE) 1996-12-17 US disclosed
US-5506246-A Method for treating depression using substituted aminomethyltetralins and their heterocyclic analogues BAYER AKTIENGESELLSCHAFT (DE) 1996-04-09 US disclosed
US-5300523-A Binding serotonin receptors, treating nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1994-04-05 US disclosed
US-5137901-A For binding 5-HT 1 receptors; treating central nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1992-08-11 US disclosed