SCHEMBL8969504

SCHEMBL8969504

Clc1ccc2c(c1)CN1C(=N2)C2CCC1C2

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
CTSD P07339 6/20 0.38
HTR2C P28335 5/20 0.33
HTR2A P28223 4/20 0.33
HTR2B P41595 3/20 0.33
HRH3 Q9Y5N1 2/20 0.32
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
AVPR1A P37288 1/20 0.31
KCNH2 Q12809 1/20 0.31
HRH1 P35367 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969499 0.89 CTSD (0.49) ACHECTSDHTR2CHTR2AHTR2B
SCHEMBL8969764 0.83 PDE3B (0.34) PDE3BPDE3AHTR2CHTR2AHTR2B
SCHEMBL8968314 0.83 PDE3B (0.40) ACHEPDE3BPDE3ACTSDHTR2C
SCHEMBL8970140 0.83 CTSD (0.32) CTSD
SCHEMBL8968679 0.81 CTSD (0.47) ACHECTSDHTR2CHTR2AHTR2B
SCHEMBL8968874 0.80 CTSD (0.41) CTSDHTR2CHTR2AHTR2BHRH3
SCHEMBL8969737 0.80 OPRM1 (0.31)
SCHEMBL8968239 0.78
SCHEMBL8968664 0.78 KLK7 (0.32) HTR2CHTR2ANOS1NOS2
SCHEMBL8969419 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed