SCHEMBL8969528

SCHEMBL8969528

COc1cc2c(c(OC)c1)N=C1C3CCC(C3)N1C2

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.35
PDE10A Q9Y233 1/20 0.33
DRD1 P21728 4/20 0.33
HTR1A P08908 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
ACHE P22303 1/20 0.32
CTSD P07339 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969818 0.80 PDE10A (0.33) PARP1PDE10ADRD1HTR1A
SCHEMBL8968749 0.78 CTSD (0.38) PARP1DRD1ACHECTSD
SCHEMBL8968644 0.75 DRD1 (0.33) PARP1DRD1HTR1AACHE
SCHEMBL8969723 0.69 HTR2C (0.36) HTR2CHTR2B
SCHEMBL8969213 0.66 ACHE (0.40) HTR2CHTR2BACHECTSD
SCHEMBL8970250 0.65 HTR2C (0.32) HTR2CHTR2B
SCHEMBL8968500 0.64 NOS1 (0.35)
SCHEMBL8968350 0.64
SCHEMBL8968239 0.64
SCHEMBL8969145 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed