SCHEMBL8973576

SCHEMBL8973576

O=C(O)CNS(=O)(=O)c1cc2ccc(Cl)cc2cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.45
ALDH1A1 P00352 2/20 0.41
APEX1 P27695 1/20 0.40
POLB P06746 1/20 0.40
ATM Q13315 1/20 0.40
MAPK1 P28482 1/20 0.40
PKLR P30613 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GAA P10253 2/20 0.39
MMP1 P03956 1/20 0.39
MMP12 P39900 1/20 0.39
ITGA1 P56199 1/20 0.39
KDM4E B2RXH2 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8789596 0.84 MAPK1 (0.55) MAPTALDH1A1POLBMAPK1HPGD
SCHEMBL3905853 0.81 APEX1 (0.57) ALDH1A1APEX1GAAMMP1MMP12
SCHEMBL31135459 0.74 CA1 (0.46) MAPTALDH1A1APEX1ATMPKLR
SCHEMBL8973003 0.72 TRPV4 (0.44) ALDH1A1HPGDITGA1L3MBTL1
SCHEMBL6846253 0.71 GAA (0.52) MAPTALDH1A1POLBMAPK1HPGD
SCHEMBL7598374 0.69 NPC1 (0.47) ALDH1A1APEX1POLBMMP1
SCHEMBL11051187 0.68 KMO (0.45) MAPTALDH1A1GAAKDM4ETDP1
SCHEMBL8972679 0.68 TPSAB1 (0.50) MAPTPOLBPKLRGAAMMP1
SCHEMBL13268374 0.68 CA1 (0.49) MAPTALDH1A1POLBHSD17B10GAA
SCHEMBL15787094 0.67 APEX1 (0.62) ALDH1A1APEX1GAAMMP1MMP12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35279-E ALDOSE REDUCTASE INHIBITORS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-06-18 US disclosed
US-5202339-A Hypoglycemic, hypolipedemic agents MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1993-04-13 US disclosed
EP-0305947-B1 HYDANTOIN DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS WELL AS THEIR USE MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1992-07-29 EP disclosed
US-5004751-A Antidiabetic agents; aldoe reductase inhibitors MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-04-02 US disclosed
US-4914099-A TREATMENT OR PREVENTION OF DIABETIC COMPLICATIONS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-04-03 US disclosed
WO-1989001934-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-09 WO disclosed
EP-0305947-A1 Hydantoin derivatives, process for their preparation and pharmaceutical compositions containing the same as well as their use MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-08 EP disclosed