SCHEMBL8974335

SCHEMBL8974335

CS(=O)(=O)c1ccc(C2=CCC=C2c2ccc(C#N)cc2)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.42
LRRK2 Q5S007 1/20 0.40
SLC22A12 Q96S37 1/20 0.38
PIK3CD O00329 1/20 0.36
PIP5K1C O60331 1/20 0.36
PIK3CB P42338 1/20 0.36
PI4KA P42356 1/20 0.36
PIK3CG P48736 1/20 0.36
PI4KB Q9UBF8 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
CTSC P53634 1/20 0.35
GPR119 Q8TDV5 2/20 0.35
CTSK P43235 1/20 0.35
MAP4K4 O95819 2/20 0.34
HSD11B1 P28845 2/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974661 0.86 CA1 (0.45) PTGS2CA12CA1CA2CA9
SCHEMBL9117303 0.83 PTGS2 (0.45) PTGS2LRRK2SLC22A12PIK3CDPIP5K1C
SCHEMBL8973871 0.83 RORC (0.41) PTGS2PIK3CDPIP5K1CPIK3CBPI4KA
SCHEMBL8974374 0.83 PIK3CD (0.39) PTGS2LRRK2PIK3CDPIP5K1CPIK3CB
SCHEMBL8974603 0.82 FAAH (0.41) PTGS2PIK3CDPIP5K1CPIK3CBPI4KA
SCHEMBL8974182 0.82 PTGS2 (0.41) PTGS2PIK3CDPIP5K1CPIK3CBPI4KA
SCHEMBL9117711 0.81 LRRK2 (0.41) PTGS2LRRK2SLC22A12PIK3CDPIP5K1C
SCHEMBL9118015 0.81 LRRK2 (0.41) PTGS2LRRK2SLC22A12PIK3CDPIP5K1C
SCHEMBL8974143 0.80 PTGS2 (0.63) PTGS2CA12CA1CA2CA9
SCHEMBL8974709 0.78 PTGS2 (0.42) PTGS2SLC22A12PIK3CDPIP5K1CPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed