SCHEMBL8985381

SCHEMBL8985381

O=[N+]([O-])c1ccc(-c2ccsc2-c2ccc(F)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 11/20 0.60
PTGS2 P35354 7/20 0.60
MAPK14 Q16539 2/20 0.58
HSPB1 P04792 1/20 0.47
GCGR P47871 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10843937 0.83 MAPK14 (0.79) PTGS1PTGS2MAPK14
SCHEMBL8985240 0.81 PTGS2 (0.69) PTGS1PTGS2
SCHEMBL8985476 0.81 PTGS1 (0.62) PTGS1PTGS2
SCHEMBL2961612 0.77 HSPB1 (0.67) PTGS1MAPK14HSPB1GCGRPOLB
SCHEMBL27458731 0.77 PTGS1 (0.46) PTGS1PTGS2MAPK14HSPB1POLB
Water SCHEMBL4218173 0.75 HSPB1 (0.64) PTGS1MAPK14HSPB1GCGRPOLB
SCHEMBL536 0.75 HSPB1 (0.75) HSPB1POLB
SCHEMBL7026994 0.75 HSPB1 (0.75) HSPB1POLB
SCHEMBL7788130 0.75 PTGS2 (0.73) PTGS1PTGS2MAPK14
SCHEMBL9259229 0.75 PTGS2 (1.00) PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5571810-A ANTIINFLAMMATORY AGENTS, ANALGESICS, COLLAGEN DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-11-05 US disclosed
EP-0593761-A1 NEW THIOPHENE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed
WO-1991019708-A1 NEW THIOPHENE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-26 WO disclosed