SCHEMBL8991084

SCHEMBL8991084

CCOCn1c(N)c(C#N)c2c(NC)ncnc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 8/20 0.42
DYRK1A Q13627 1/20 0.35
HSPA8 P11142 1/20 0.34
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
YTHDC1 Q96MU7 1/20 0.31
MAPK13 O15264 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
MAPK14 Q16539 1/20 0.31
MAPK8 P45983 1/20 0.31
MAPK9 P45984 1/20 0.31
GRK6 P43250 1/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
GLA P06280 2/20 0.31
GAA P10253 2/20 0.31
HPGD P15428 2/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8991164 0.87 LRRK2 (0.40) LRRK2DYRK1AHSPA8CDK5CDK5R1
SCHEMBL7697510 0.86 LRRK2 (0.58) LRRK2DYRK1AHSPA8CDK5CDK5R1
SCHEMBL8991180 0.84 LRRK2 (0.43) LRRK2KDM4EALDH1A1GLAGAA
SCHEMBL8991004 0.77 YTHDC1 (0.31) YTHDC1EGFRSRC
SCHEMBL8991158 0.77 KMT2A (0.49) LRRK2KDM4EALDH1A1GLAGAA
SCHEMBL8991163 0.77 YTHDC1 (0.31) YTHDC1EGFRSRC
SCHEMBL8990982 0.76 GAA (0.42) LRRK2KDM4EALDH1A1GLAGAA
SCHEMBL8991316 0.76 ALDH1A1 (0.55) LRRK2KDM4EALDH1A1GLAGAA
SCHEMBL8991012 0.74 XDH (0.33)
SCHEMBL8991176 0.74 XDH (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5543413-A VIRAL ACTIVITY AGAINST HUMAN CYTOMEGALOVIRUS AND HERPES SIMPLEX VIRUS REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 1996-08-06 US disclosed