SCHEMBL8992825

SCHEMBL8992825

COc1cc(COC2CCCCO2)ccc1C(O)c1cccc(C)c1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.37
CREBBP Q92793 2/20 0.35
ICAM1 P05362 1/20 0.35
SELE P16581 1/20 0.35
ALDH1A1 P00352 1/20 0.34
EP300 Q09472 1/20 0.33
PDE4B Q07343 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
PTPN1 P18031 1/20 0.32
ITGB1 P05556 1/20 0.32
ITGA4 P13612 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8993283 0.90 TACR1 (0.40) TACR1CREBBPICAM1SELENPC1
SCHEMBL8992789 0.83 TACR1 (0.40) TACR1ICAM1SELENPC1RAB9A
SCHEMBL8992790 0.80 TACR1 (0.43) TACR1CREBBPICAM1SELEEP300
SCHEMBL8992804 0.78 DHFR (0.39) TACR1CREBBPICAM1SELENPC1
SCHEMBL93016 0.74 SMN1; SMN2 (0.47) CREBBPICAM1SELEALDH1A1PDE4B
SCHEMBL18410184 0.74 ICAM1 (0.40) CREBBPICAM1SELEEP300NPC1
SCHEMBL18410186 0.73 NPC1 (0.40) CREBBPICAM1SELEALDH1A1EP300
SCHEMBL27343854 0.73 CREBBP (0.38) TACR1CREBBPICAM1SELEEP300
SCHEMBL27287536 0.73 TACR1 (0.43) TACR1CREBBPEP300NPC1RAB9A
SCHEMBL8632096 0.71 ALDH1A1 (0.50) TACR1ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed