SCHEMBL8992789

SCHEMBL8992789

COc1cccc(C(O)c2ccc(COC3CCCCO3)cc2C)c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
HPGD P15428 2/20 0.38
LMNA P02545 1/20 0.38
BRD4 O60885 1/20 0.37
POLB P06746 1/20 0.36
FFAR1 O14842 3/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ICAM1 P05362 1/20 0.35
SELE P16581 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8993283 0.90 TACR1 (0.40) TACR1NPC1RAB9AHPGDLMNA
SCHEMBL8992790 0.88 TACR1 (0.43) TACR1SLC6A3ICAM1SELE
SCHEMBL8992825 0.83 TACR1 (0.37) TACR1NPC1RAB9ASLC6A2SLC6A4
SCHEMBL8632096 0.80 ALDH1A1 (0.50) TACR1NPC1RAB9ALMNAPOLB
SCHEMBL8992916 0.78 DHFR (0.46) TACR1NPC1RAB9AHPGDLMNA
SCHEMBL8992732 0.76 BRD4 (0.40) BRD4FFAR1
SCHEMBL8992895 0.75 AOC3 (0.45) BRD4
SCHEMBL93016 0.74 SMN1; SMN2 (0.47) NPC1RAB9ATDP1ICAM1SELE
SCHEMBL27343854 0.73 CREBBP (0.38) TACR1LMNASLC6A3ICAM1SELE
SCHEMBL8321396 0.72 NPC1 (0.50) TACR1NPC1RAB9AICAM1SELE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed