SCHEMBL8992841

SCHEMBL8992841

COc1cc(Cc2ccc(CC#N)cc2)cc(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CALM1 P0DP23 5/20 0.50
PKM P14618 1/20 0.46
FGFR3 P22607 1/20 0.44
LTA4H P09960 1/20 0.44
CYP19A1 P11511 1/20 0.43
FLT3 P36888 1/20 0.41
AKR1B1 P15121 1/20 0.41
ALDH1A1 P00352 1/20 0.39
PIK3CD O00329 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37
CA2 P00918 1/20 0.37
NPC1 O15118 1/20 0.37
THRB P10828 1/20 0.37
RAB9A P51151 1/20 0.37
SAE1 Q9UBE0 1/20 0.37
UBA2 Q9UBT2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8992958 0.87 LTA4H (0.59) PKMLTA4HFLT3ALDH1A1CA2
SCHEMBL27327790 0.86 CYP19A1 (0.61) CALM1PKMFGFR3CYP19A1FLT3
SCHEMBL8992947 0.85 LTA4H (0.49) LTA4H
SCHEMBL1046247 0.85 ALDH1A1 (0.50) CALM1PKMFGFR3CYP19A1FLT3
SCHEMBL31739223 0.82 MAOA (0.51) CALM1LTA4HCYP19A1AKR1B1RAB9A
SCHEMBL9203057 0.81 ALDH1A1 (0.43) CALM1PKMFGFR3CYP19A1FLT3
3-Methoxyphenylacetonitrile SCHEMBL103029 0.81 PKM (0.61) CALM1PKMLTA4HFLT3ALDH1A1
3-Methoxyphenylacetonitrile SCHEMBL29253102 0.79 PKM (0.59) PKMLTA4HFLT3ALDH1A1CA2
3-Methoxyphenylacetonitrile SCHEMBL27728444 0.79 PKM (0.59) CALM1PKMLTA4HFLT3ALDH1A1
SCHEMBL5252553 0.78 ALDH1A1 (0.65) CALM1LTA4HCYP19A1AKR1B1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed