SCHEMBL8992958

SCHEMBL8992958

COc1ccc(Cc2ccc(CC#N)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.59
PKM P14618 1/20 0.56
SAE1 Q9UBE0 1/20 0.47
UBA2 Q9UBT2 1/20 0.47
FLT3 P36888 1/20 0.47
IDO1 P14902 3/20 0.47
ALDH1A1 P00352 3/20 0.44
GAA P10253 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
AGXT P21549 2/20 0.44
TAAR1 Q96RJ0 1/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
CYP2D6 P10635 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
3-Methoxyphenylacetonitrile SCHEMBL103029 0.94 PKM (0.61) LTA4HPKMFLT3IDO1ALDH1A1
3-Methoxyphenylacetonitrile SCHEMBL29253102 0.92 PKM (0.59) LTA4HPKMFLT3IDO1ALDH1A1
3-Methoxyphenylacetonitrile SCHEMBL27728444 0.92 PKM (0.59) LTA4HPKMFLT3IDO1ALDH1A1
3-Methoxyphenylacetonitrile SCHEMBL28155308 0.90 PKM (0.58) LTA4HPKMFLT3IDO1ALDH1A1
SCHEMBL5004118 0.88 FLT3 (0.57) LTA4HPKMFLT3IDO1ALDH1A1
SCHEMBL8992841 0.87 CALM1 (0.50) LTA4HPKMSAE1UBA2FLT3
3-Methoxyphenylacetonitrile SCHEMBL7135147 0.86 LTA4H (0.62) LTA4HPKMFLT3IDO1ALDH1A1
SCHEMBL3520397 0.83 APP (0.61) PKMIDO1ALDH1A1AGXTMAOB
SCHEMBL6933353 0.83 PKM (0.52) LTA4HPKMFLT3IDO1ALDH1A1
SCHEMBL8992947 0.83 LTA4H (0.49) LTA4HIDO1AGXTTAAR1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1036919-C Pyrazole condensed ring derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMA CO LTD (JP) 1998-01-07 CN disclosed
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed