SCHEMBL8992896

SCHEMBL8992896

Nc1n[nH]cc1-c1ccc(Cc2ccc3c(c2)OCO3)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.47
ALDH1A1 P00352 1/20 0.44
HSD17B10 Q99714 1/20 0.44
LTB4R Q15722 1/20 0.43
TAAR1 Q96RJ0 3/20 0.43
SLC6A4 P31645 2/20 0.42
ADORA2A P29274 1/20 0.42
FYN P06241 1/20 0.41
ADORA1 P30542 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CHEK2 O96017 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL108109 0.76 TAAR1 (0.62) ALDH1A1TAAR1SLC6A4SLC6A2SLC6A3
SCHEMBL8993116 0.75 LTA4H (0.45) MPOLTB4RCYP3A4CYP2D6
SCHEMBL109195 0.74 TAAR1 (0.64) ALDH1A1TAAR1SLC6A4SLC6A2SLC6A3
SCHEMBL8992834 0.73 LTA4H (0.53) MPOALDH1A1TAAR1CYP3A4CHEK2
SCHEMBL9036923 0.72 PTGS2 (0.51) ALDH1A1TAAR1SLC6A4CYP3A4
SCHEMBL8993151 0.72 CYP3A4 (0.57) ALDH1A1TAAR1SLC6A4SLC6A2SLC6A3
SCHEMBL8992951 0.71 LTA4H (0.57) LTB4RTAAR1ADORA1
SCHEMBL8993059 0.70 CHEK2 (0.43) ALDH1A1HSD17B10LTB4RCYP3A4CHEK2
SCHEMBL1422874 0.70 ALDH1A1 (0.58) ALDH1A1TAAR1SLC6A4SLC6A2SLC6A3
SCHEMBL15599268 0.69 LTB4R (0.50) MPOALDH1A1HSD17B10LTB4RTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed