SCHEMBL8993128

SCHEMBL8993128

COc1cccc(Cc2ccc(COC3CCCCO3)cc2OC)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.46
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 1/20 0.40
CNR1 P21554 3/20 0.40
GPR55 Q9Y2T6 3/20 0.40
TACR1 P25103 1/20 0.40
CNR2 P34972 4/20 0.40
ABCB1 P08183 1/20 0.40
ICAM1 P05362 1/20 0.38
SELE P16581 1/20 0.38
IDO1 P14902 2/20 0.38
AGXT P21549 2/20 0.38
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8992804 0.90 DHFR (0.39) DHFRNPC1RAB9ACNR1TACR1
SCHEMBL8992916 0.90 DHFR (0.46) DHFRNPC1RAB9AALDH1A1CNR1
SCHEMBL8632096 0.88 ALDH1A1 (0.50) DHFRNPC1RAB9AALDH1A1TACR1
SCHEMBL8993283 0.78 TACR1 (0.40) NPC1RAB9ATACR1ICAM1SELE
SCHEMBL18410186 0.76 NPC1 (0.40) NPC1RAB9AALDH1A1ICAM1SELE
SCHEMBL8993256 0.76 KDM4C (0.41) DHFRTACR1ICAM1SELE
SCHEMBL8321396 0.75 NPC1 (0.50) NPC1RAB9ATACR1ICAM1SELE
SCHEMBL93016 0.75 SMN1; SMN2 (0.47) NPC1RAB9AALDH1A1ICAM1SELE
SCHEMBL5423197 0.74 NPC1 (0.52) DHFRNPC1RAB9AALDH1A1TACR1
SCHEMBL18410184 0.74 ICAM1 (0.40) NPC1RAB9AICAM1SELE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed