SCHEMBL8993203

SCHEMBL8993203

COc1cccc(Cc2ccc(C[Si](C)(C)C(C)(C)C)cc2C)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.44
GPR55 Q9Y2T6 2/20 0.44
CNR1 P21554 2/20 0.44
DHFR P00374 1/20 0.43
FGFR1 P11362 1/20 0.41
FGFR4 P22455 1/20 0.41
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
HTR1B P28222 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
IDH1 O75874 1/20 0.39
LTA4H P09960 1/20 0.39
IDO1 P14902 1/20 0.38
AGXT P21549 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
NMT1 P30419 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8992799 0.83 IDO1 (0.46) CNR2GPR55CNR1DHFRFGFR1
SCHEMBL8993136 0.79 CNR2 (0.46) CNR2GPR55CNR1DHFRFGFR1
SCHEMBL8993225 0.79 IDH1 (0.47) CNR2GPR55CNR1DHFRFGFR1
SCHEMBL5648684 0.77 CNR2 (0.52) CNR2GPR55CNR1DHFRFGFR1
SCHEMBL8992807 0.75 CNR2 (0.46) CNR2GPR55CNR1DHFRFGFR1
SCHEMBL5646180 0.74 ANO1 (0.50) CNR2GPR55CNR1DHFRFGFR1
SCHEMBL8992916 0.73 DHFR (0.46) CNR2GPR55CNR1DHFRIDO1
Hydrochloric Acid SCHEMBL27513621 0.71 IDO1 (0.36) CHRM2CHRM1CHRM3IDO1AGXT
SCHEMBL28842002 0.70 LTA4H (0.55) CNR2LTA4HIDO1
SCHEMBL21365120 0.69 CA2 (0.52) CNR2GPR55CNR1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed