SCHEMBL8994243

SCHEMBL8994243

O=C1C=CC2=Nc3ccccc3CCC2=C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.49
NOS1 P29475 1/20 0.49
NOS2 P35228 1/20 0.49
NPC1 O15118 5/20 0.39
RAB9A P51151 4/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPT P10636 1/20 0.39
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
HPGD P15428 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
MAPK13 O15264 1/20 0.33
MAPK12 P53778 1/20 0.33
MAPK11 Q15759 1/20 0.33
MAPK14 Q16539 1/20 0.33
CES1 P23141 1/20 0.33
CYP2A6 P11509 1/20 0.32
ACHE P22303 5/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7873710 0.85 NOS3 (0.38) NOS3NOS1NOS2NPC1RAB9A
SCHEMBL8994244 0.78 PDE3B (0.42) ALDH1A1PDE3BPDE3ALMNACYP3A4
SCHEMBL14730907 0.78 ACHE (0.36) PDE3BPDE3AACHESRD5A1
SCHEMBL9279571 0.74 KDM4E (0.45) NOS3NOS1NOS2NPC1RAB9A
SCHEMBL14141233 0.69 NOS3 (0.54) NOS3NOS1NOS2RAB9AOPRM1
SCHEMBL2075410 0.66 NOS3 (1.00) NOS3NOS1NOS2NPC1RAB9A
Hydrochloric Acid SCHEMBL8324907 0.65 NOS3 (0.96) NOS3NOS1NOS2NPC1RAB9A
SCHEMBL30804593 0.65 MAOA (0.38) NPC1RAB9AALDH1A1MAPTHPGD
SCHEMBL3348606 0.65 MAOA (0.38) NPC1RAB9AALDH1A1MAPTHPGD
SCHEMBL19968930 0.64 NPSR1 (0.35) HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0542019-B1 8-Hydroxy-2H-dibenz(b,f) azepin-2 one dyes BAYER AG (US) 1996-08-14 EP disclosed
EP-0542019-A1 8-Hydroxy-2H-dibenz(b,f) azepin-2 one dyes Bayer Corporation (US) 1993-05-19 EP disclosed
US-5208326-A 8-HYDROXY-2H-DIBENZ(B,F)AZEPIN-2-ONE DYES MILES INC. (US) 1993-05-04 US disclosed