SCHEMBL8995008

SCHEMBL8995008

CC(=O)/N=C(\N)c1ccc(OCCCCCOc2ccc(C(=O)N(c3ccccc3)C(C)C)c(Cl)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 7/20 0.39
THRA P10827 1/20 0.39
THRB P10828 1/20 0.39
LTB4R Q15722 2/20 0.37
NPC1 O15118 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37
S1PR3 Q99500 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LTB4R2 Q9NPC1 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
MAOB P27338 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8748025 0.91 RAB9A (0.47) NR1H4THRATHRBLTB4RNPC1
SCHEMBL8748028 0.91 RAB9A (0.47) NR1H4THRATHRBLTB4RNPC1
SCHEMBL8995004 0.87 LTB4R (0.50) LTB4RLTB4R2
SCHEMBL8994927 0.87 LTB4R (0.47) THRATHRBLTB4RNPC1PKM
Hydrochloric Acid SCHEMBL8994888 0.86 LTB4R (0.49) LTB4RLTB4R2
SCHEMBL8995015 0.83 ATM (0.40) NR1H4THRATHRBMTNR1AMTNR1B
SCHEMBL8995022 0.82 CA1 (0.41) NR1H4THRATHRBMAOB
SCHEMBL8748089 0.81 THRA (0.42) NR1H4THRATHRBNPC1
Hydrochloric Acid SCHEMBL8994900 0.81 CA1 (0.41) NR1H4THRATHRBMAOB
SCHEMBL8747936 0.81 GAA (0.47) LTB4RNPC1RAB9ATDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5488160-A LEUKOTRIENE B4 RECEPTOR ANTAGONIST AS ANTIINFLAMMATORY AGENTS CIBA-GEIGY CORPORATION (US) 1996-01-30 US disclosed