SCHEMBL8997214

SCHEMBL8997214

C=CC(CCC1CNc2nc(N)nc(N)c21)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ATIC P31939 2/20 0.49
GART P22102 6/20 0.48
SOST Q9BQB4 1/20 0.46
MTHFD2 P13995 2/20 0.46
MTHFD1 P11586 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997198 0.89 ATIC (0.48) ATICGART
SCHEMBL8997170 0.88 DHFR (0.55) ATICGART
SCHEMBL9758306 0.88 DHFR (0.55) ATICGART
SCHEMBL8997253 0.86 DHFR (0.58) ATICGART
SCHEMBL9397716 0.85 DHFR (0.53) ATICGART
SCHEMBL9227822 0.85 DHFR (0.52) ATICGART
SCHEMBL9758337 0.84 DHFR (0.60) ATICGART
SCHEMBL8997146 0.84 ATIC (0.50) ATICGART
SCHEMBL8997257 0.83 GART (0.61) ATICGART
SCHEMBL9041817 0.83 MTHFD1 (0.59) ATICGARTSOSTMTHFD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5296600-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-22 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
EP-0334636-A2 Pyrrolopyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-09-27 EP disclosed