SCHEMBL8997153

SCHEMBL8997153

COC(=O)c1ccc(CCCC2CNc3nc(N)n(COC(C)C)c(=O)c32)cc1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 2/20 0.36
CYP4F2 P78329 1/20 0.36
EP300 Q09472 8/20 0.35
GART P22102 1/20 0.34
TLR7 Q9NYK1 1/20 0.33
ATIC P31939 2/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
EHMT2 Q96KQ7 1/20 0.33
DHODH Q02127 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997195 0.95 ATIC (0.35) CYP4A11CYP4F2EP300GARTTLR7
SCHEMBL8997209 0.76 CYP4A11 (0.43) CYP4A11CYP4F2EP300GARTTLR7
SCHEMBL8997279 0.70 DHFR (0.40) CYP4A11CYP4F2TLR7ATICMAPT
SCHEMBL9844790 0.70 EP300 (0.38) CYP4A11CYP4F2EP300MAPTTHRB
SCHEMBL8997437 0.68 DHFR (0.44) CYP4A11GART
SCHEMBL9844748 0.67 DRD2 (0.39) EP300TLR7MAPTTHRBMEN1
SCHEMBL9844763 0.64 NPC1 (0.36) TLR7MAPTMEN1KMT2A
SCHEMBL9844745 0.64 MAPT (0.35) TLR7MAPTMEN1KMT2A
SCHEMBL7505320 0.62 CYP4A11 (0.60) CYP4A11CYP4F2MAPTTHRB
SCHEMBL14967206 0.62 CYP4A11 (0.58) CYP4A11CYP4F2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5296600-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-22 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0334636-A2 Pyrrolopyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-09-27 EP disclosed