SCHEMBL9001771

SCHEMBL9001771

Nc1nc2c(c(=O)[nH]1)C(CCc1ccc(C(=O)O)cc1)CC2

nearest known ligand 0.68

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ATIC P31939 4/20 0.41
GART P22102 5/20 0.40
TYMS P04818 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001819 0.85 ATIC (0.37) ATICGARTTYMS
SCHEMBL7831766 0.81 ATIC (0.51) ATICGARTTYMS
SCHEMBL8566937 0.81 MTR (0.44)
SCHEMBL8567466 0.74 MTR (0.41)
SCHEMBL27891667 0.71 PTGER4 (0.47) ATICTYMS
SCHEMBL7812453 0.71 GART (0.69) ATICGARTTYMS
SCHEMBL9038667 0.68 GART (0.64) ATICGART
SCHEMBL9215453 0.67 GART (0.52) ATICGARTTYMS
SCHEMBL7612737 0.66 GART (0.65) ATICGARTTYMS
SCHEMBL7742870 0.66 DHFR (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed