SCHEMBL7742870

SCHEMBL7742870

Nc1nc(N)c2c(n1)OCC2CCc1ccc(C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
ATM Q13315 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MBOAT4 Q96T53 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TAAR1 Q96RJ0 1/20 0.36
NOS1 P29475 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6427011 0.87 DHFR (0.43) DHFRKMT2AALDH1A1HPGDHSD17B10
SCHEMBL8566937 0.80 MTR (0.44) DHFRPOLBMAPTKMT2AATM
SCHEMBL8567466 0.74 MTR (0.41) DHFRPOLBMAPTKMT2AATM
SCHEMBL8562117 0.68 MTR (0.44) DHFR
SCHEMBL7660756 0.66 P2RX3 (0.47) DHFRPOLBMAPTKMT2AATM
SCHEMBL9001771 0.66 ATIC (0.41)
SCHEMBL27580519 0.66 ALDH1A1 (0.48) MAPTKMT2AALDH1A1
SCHEMBL9341089 0.64 CYP2D6 (0.53) DHFRPOLBMAPTKMT2AATM
SCHEMBL9338914 0.64 CYP2D6 (0.56) DHFRPOLBMAPTKMT2AATM
SCHEMBL8997177 0.64 NOS1 (0.39) DHFRMAPTKMT2AALDH1A1NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420370-B1 ANTITUMOR, ANTIBIOTIC, ANTIMALARIAL, ANTIFUNGAL OR ANTIPROTOZOAL AGENTS, OR AS SYNERGISTIC AGENTS ENZYME INHIBITORS DUQUESNE UNIVERSITY OF THE HOLY GHOST 2002-07-16 US disclosed