SCHEMBL9001972

SCHEMBL9001972

O=C(O)CN(CCN(CCN(CC(=O)O)CC(=O)O)[C@@H](Cc1ccc(I)cc1)C(=O)O)CC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.40
EYA2 O00167 1/20 0.40
APP P05067 1/20 0.40
ACE P12821 1/20 0.40
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
CHRM2 P08172 1/20 0.39
ADRA2A P08913 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
DRD1 P21728 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
CYP2C19 P33261 1/20 0.39
ADRA1A P35348 1/20 0.39
DRD3 P35462 1/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
SLC6A3 Q01959 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7513236 0.86 TDP1 (0.40) TDP1EYA2APPACEKDM4E
SCHEMBL7598191 0.83 SLC7A5 (0.44) TDP1EYA2APPACEKDM4E
SCHEMBL29588115 0.82 CYP1A2 (0.43) TDP1EYA2APPACEKDM4E
SCHEMBL7596061 0.82 CYP1A2 (0.43) TDP1EYA2APPACEKDM4E
SCHEMBL9435308 0.82 TDP1 (0.39) TDP1EYA2APPACEKDM4E
SCHEMBL5252487 0.82 TDP1 (0.39) TDP1EYA2APPACEKDM4E
SCHEMBL7514789 0.81 ALOX15 (0.41) ALOX15TSHR
SCHEMBL7630147 0.80 SLC7A5 (0.39) CA1CA2CA4
SCHEMBL8386941 0.80 ITGB3 (0.48) TDP1
SCHEMBL7950553 0.80 ALDH1A1 (0.44) CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731784-A1 ARYL HALIDE SUBSTITUTED METALLIC COMPLEXES, PHARMACEUTICALS CONTAINING THESE COMPLEXES, THEIR USE FOR DIAGNOSTIC PURPOSES, AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1996-09-18 EP disclosed
WO-1995015306-A1 ARYL HALIDE SUBSTITUTED METALLIC COMPLEXES, PHARMACEUTICALS CONTAINING THESE COMPLEXES, THEIR USE FOR DIAGNOSTIC PURPOSES, AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1995-06-08 WO disclosed