SCHEMBL9002071

SCHEMBL9002071

O=C(Nc1cccc2ccccc12)OCCSc1cccc2nccn12

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
HPGD P15428 2/20 0.47
LMNA P02545 5/20 0.44
NPC1 O15118 1/20 0.43
MAPT P10636 4/20 0.43
KDM4E B2RXH2 1/20 0.42
APOBEC3A P31941 1/20 0.42
HTT P42858 1/20 0.42
APOBEC3G Q9HC16 1/20 0.42
TP53 P04637 3/20 0.41
THRB P10828 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002036 0.84 LMNA (0.48) ALDH1A1LMNANPC1MAPTTP53
SCHEMBL9001935 0.79 QPCT (0.50) ALDH1A1HPGDLMNANPC1MAPT
SCHEMBL9002225 0.78 PKM (0.40) ALDH1A1LMNAMAPTHTTPKM
SCHEMBL9001998 0.77 SMN1; SMN2 (0.34) MAPK1
SCHEMBL8581462 0.77 PTGS2 (0.36) ALDH1A1HPGDNPC1MAPTKDM4E
SCHEMBL9002235 0.77 SMN1; SMN2 (0.42) ALDH1A1HPGDNPC1MAPTKDM4E
SCHEMBL9002520 0.76 ACHE (0.43) HPGDHTTPOLB
Hydrochloric Acid SCHEMBL9002227 0.73 HPGD (0.49) ALDH1A1HPGDLMNANPC1MAPT
SCHEMBL9001857 0.73 HPGD (0.34) HPGDNPC1HTTTP53L3MBTL1
SCHEMBL9001983 0.71 ALDH1A1 (0.52) ALDH1A1HPGDLMNANPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed