SCHEMBL9012482

SCHEMBL9012482

CCCCCC(=O)N=C(NC(=O)OC(C)(C)C)n1cccn1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 3/20 0.38
CNR2 P34972 1/20 0.31
CTSK P43235 3/20 0.31
CYP3A4 P08684 1/20 0.30
PCSK9 Q8NBP7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4249587 0.86 NOS1 (0.36) NOS1CTSK
SCHEMBL4249589 0.86 NOS1 (0.36) NOS1CTSK
SCHEMBL9012507 0.83 NOS1 (0.43) NOS1
SCHEMBL8196578 0.83 NOS1 (0.34) NOS1
SCHEMBL14135 0.83 RAB9A (0.32) NOS1PCSK9
SCHEMBL8121 0.83 RAB9A (0.32) NOS1PCSK9
SCHEMBL13221 0.83 RAB9A (0.32) NOS1PCSK9
SCHEMBL2703386 0.83 NOS1 (0.50) NOS1CNR2PCSK9
SCHEMBL24177802 0.83 PCSK9 (0.33) NOS1PCSK9
SCHEMBL8199304 0.83 NOS1 (0.34) NOS1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743320-A2 Acyl guanidine and amidine prodrugs BRISTOL-MYERS SQUIBB COMPANY (US) 1996-11-20 EP disclosed