SCHEMBL9013871

SCHEMBL9013871

CCCCCCCCCCCCC(CCC)Nc1ccc(OC2CCNCC2)c(C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.36
PDE4B Q07343 2/20 0.36
PDE4C Q08493 2/20 0.36
PDE4D Q08499 2/20 0.36
TOP2A P11388 1/20 0.35
BCL9 O00512 1/20 0.34
CTNNB1 P35222 1/20 0.34
SLC6A4 P31645 2/20 0.33
P2RX3 P56373 1/20 0.33
HRH1 P35367 2/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
GNAI3 P08754 1/20 0.32
GNAO1 P09471 1/20 0.32
GNAI1 P63096 1/20 0.32
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
ESR1 P03372 1/20 0.31
HTR1A P08908 1/20 0.31
SLC6A2 P23975 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9022461 0.99 TOP2A (0.35) PDE4APDE4BPDE4CPDE4DTOP2A
SCHEMBL9022423 0.83 SLC6A4 (0.38) PDE4APDE4BPDE4CPDE4DTOP2A
SCHEMBL9013880 0.81 ABL1 (0.40) TOP2ABCL9CTNNB1SLC6A4GNAI3
SCHEMBL9022813 0.81 ABL1 (0.40) TOP2ABCL9CTNNB1SLC6A4GNAI3
SCHEMBL9023282 0.80 BCL9 (0.39) TOP2ABCL9CTNNB1SLC6A4HRH1
Hydrochloric Acid SCHEMBL9013913 0.76 GNAI3 (0.46) TOP2ABCL9CTNNB1GNAI3GNAO1
SCHEMBL21139473 0.71 TAS1R3 (0.56) TAS1R3TAS1R1
SCHEMBL171093 0.68 HTR2C (0.47) SLC6A4HRH1HTR2CHTR2BHTR1A
SCHEMBL9022486 0.67 HRH1 (0.47) HRH1
SCHEMBL9023137 0.66 RAB9A (0.45) PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5580883-A INHIBITING DEGENERATION AND NECROCYTOSIS OF CEREBRAL NERVE CELLS CAUSED BY OXIDATIVE STRESS INDUCING GLUTAMIC ACID IN MAMMALS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-03 US disclosed
EP-0449195-B1 Aminobenzene compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-05-08 EP disclosed
EP-0449195-A2 Aminobenzene compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-10-02 EP disclosed