SCHEMBL9014407

SCHEMBL9014407

N#Cc1ccc2c(c1)OCCCC2CCBr

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.37
DRD3 P35462 3/20 0.37
LRRK2 Q5S007 4/20 0.35
KDM4C Q9H3R0 2/20 0.33
MAP3K5 Q99683 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
CHRNA1 P02708 1/20 0.32
CHRNG P07510 1/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
CHRND Q07001 1/20 0.32
GRM5 P41594 1/20 0.32
SLC6A4 P31645 2/20 0.31
MAOB P27338 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014733 0.90 DRD2 (0.39) DRD2DRD3PTGDR2NOS3NOS1
SCHEMBL9014727 0.76 KCNH2 (0.38)
SCHEMBL9014643 0.74 TERT (0.38) CHRNB4CHRNA3NOS3NOS1NOS2
SCHEMBL9014726 0.74 MAP3K14 (0.33)
SCHEMBL9014335 0.71 KDM4E (0.37) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9234439 0.71 DRD3 (0.37) DRD2DRD3MAOB
SCHEMBL9014788 0.71 ADRA2A (0.40) DRD2DRD3PTGDR2MAOB
SCHEMBL4138299 0.71 LRRK2 (0.42) DRD2DRD3LRRK2CHRNA1CHRNG
SCHEMBL5394460 0.71 LRRK2 (0.42) DRD2DRD3LRRK2CHRNA1CHRNG
SCHEMBL31715704 0.71 LRRK2 (0.42) DRD2DRD3LRRK2CHRNA1CHRNG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed