SCHEMBL9014335

SCHEMBL9014335

Nc1ccc2c(c1)C(CCBr)CCCO2

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
HTR1A P08908 1/20 0.35
HTR1D P28221 1/20 0.35
HTR2C P28335 1/20 0.35
MTNR1A P48039 2/20 0.31
MTNR1B P49286 2/20 0.31
CHRNB4 P30926 4/20 0.31
CHRNA3 P32297 4/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNA4 P43681 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9234439 0.83 DRD3 (0.37) KDM4EGAAMAPTHTR1AHTR1D
SCHEMBL9014788 0.83 ADRA2A (0.40) HTR1AHTR1DHTR2CMTNR1AMTNR1B
SCHEMBL9014302 0.80 HTR1A (0.47) HTR1AMTNR1AMTNR1B
SCHEMBL9014733 0.80 DRD2 (0.39) ALDH1A1
SCHEMBL9014727 0.79 KCNH2 (0.38) MTNR1AMTNR1B
SCHEMBL10408558 0.74 MAP3K14 (0.45) HTR1AMTNR1AMTNR1B
SCHEMBL10407574 0.74 ADRA2A (0.36) HTR1AMTNR1AMTNR1B
SCHEMBL10407837 0.74 DRD3 (0.39) KDM4EHTR1AHTR1DHTR2CMTNR1A
SCHEMBL8139731 0.73 MTNR1A (0.36) KDM4EGAAMAPTHTR1AHTR1D
SCHEMBL9014396 0.71 MAP3K14 (0.35) MTNR1AMTNR1BCHRNB4CHRNA3CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed