SCHEMBL9014643

SCHEMBL9014643

O=[N+]([O-])c1ccc2c(c1)OCCCC2CCBr

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TERT O14746 1/20 0.38
ALDH1A1 P00352 4/20 0.38
GAA P10253 1/20 0.38
CHRNB4 P30926 5/20 0.37
CHRNA3 P32297 5/20 0.37
HSP90AA1 P07900 1/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
ACHE P22303 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LMNA P02545 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10407545 0.82 HSP90AA1 (0.38) ALDH1A1CHRNB4CHRNA3HSP90AA1MEN1
SCHEMBL9014699 0.78 PNMT (0.40) CHRNB4CHRNA3HSP90AA1NOS3NOS1
SCHEMBL9014349 0.75 CHRNB4 (0.36) ALDH1A1CHRNB4CHRNA3ACHEMEN1
SCHEMBL9014407 0.74 DRD2 (0.37) CHRNB4CHRNA3NOS3NOS1NOS2
SCHEMBL9014727 0.74 KCNH2 (0.38) SMN1; SMN2LMNACRHBPCRHR2
SCHEMBL9014394 0.72 KCNH2 (0.64) ALDH1A1GAAMEN1KMT2ASMN1; SMN2
SCHEMBL10845095 0.70 MEN1 (0.54) TERTALDH1A1CHRNB4CHRNA3MEN1
SCHEMBL9014335 0.69 KDM4E (0.37) ALDH1A1GAACHRNB4CHRNA3KDM4E
SCHEMBL6350114 0.69 HSP90AA1 (0.47) ALDH1A1CHRNB4CHRNA3HSP90AA1MEN1
SCHEMBL6347584 0.69 HSP90AA1 (0.43) ALDH1A1CHRNB4CHRNA3HSP90AA1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed