SCHEMBL9014733

SCHEMBL9014733

N#Cc1ccc2c(c1)C(CCBr)CCCO2

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.39
DRD3 P35462 10/20 0.39
ABCB1 P08183 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
ABCC9 O60706 2/20 0.33
ABCC8 Q09428 2/20 0.33
KCNJ11 Q14654 2/20 0.33
KCNJ8 Q15842 2/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
LMNA P02545 1/20 0.33
HCRTR2 O43614 1/20 0.33
ALDH1A1 P00352 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014407 0.90 DRD2 (0.37) DRD2DRD3PTGDR2NOS3NOS1
SCHEMBL9014335 0.80 KDM4E (0.37) ALDH1A1
SCHEMBL9014788 0.80 ADRA2A (0.40) DRD2DRD3PTGDR2HCRTR2
SCHEMBL9234439 0.80 DRD3 (0.37) DRD2DRD3CYP1A2CYP2D6CYP2C19
SCHEMBL9014302 0.76 HTR1A (0.47) DRD2DRD3
SCHEMBL9585693 0.76 DRD2 (0.40) DRD2DRD3ABCB1ABCC9ABCC8
SCHEMBL9014727 0.76 KCNH2 (0.38) LMNA
SCHEMBL8402481 0.75 DRD2 (0.47) DRD2DRD3ABCB1CYP1A2CYP2D6
SCHEMBL6215060 0.72 HTR1A (0.57) DRD2DRD3ABCB1HCRTR2
SCHEMBL29243618 0.71 DRD2 (0.42) DRD2DRD3ABCB1NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed