SCHEMBL9014787

SCHEMBL9014787

COc1cccc2c1C(CCBr)CCCO2

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.39
CTNNB1 P35222 1/20 0.36
WNT3A P56704 1/20 0.36
MAP3K14 Q99558 1/20 0.35
DRD2 P14416 1/20 0.34
DRD1 P21728 1/20 0.34
HTR1B P28222 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
CTSG P08311 1/20 0.34
KLK7 P49862 1/20 0.34
KLK14 Q9P0G3 1/20 0.34
KLK5 Q9Y337 1/20 0.34
ABCB1 P08183 1/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014383 0.85 MTNR1A (0.40) CTNNB1WNT3AMAP3K14
SCHEMBL9014723 0.81 MAP3K14 (0.36) MAP3K14
SCHEMBL9014396 0.80 MAP3K14 (0.35) MAP3K14
SCHEMBL9015271 0.80 MAP3K14 (0.35) MAP3K14CTSGKLK7KLK14KLK5
SCHEMBL9014726 0.76 MAP3K14 (0.33) MAP3K14
SCHEMBL9014349 0.74 CHRNB4 (0.36) MAP3K14
SCHEMBL9014647 0.74 KCNH2 (0.68) HTR1ADRD2KCNH2
SCHEMBL9014337 0.74 MTNR1A (0.42) MAP3K14
Hydrochloric Acid SCHEMBL29960788 0.74 HTR1A (0.54) HTR1ACTNNB1WNT3AMAP3K14HTR2A
SCHEMBL9014727 0.73 KCNH2 (0.38) HTR2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed